O zolpidem tem meia-vida curta, ou seja, é absorvido rapidamente pelo organismo e perde o efeito em poucas horas — em média, quatro. Esse metabolismo acelerado faz com que o corpo se acostume rapidamente, e o usuário acabe aumentando a dose para tentar reproduzir o efeito inicial. Quanto menor a meia-vida de um medicamento, maior tende a ser o seu potencial de dependência.
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